Webb1 maj 1992 · With P1-Asn, reversible inhibition could be demonstrated directly upon dilution of preformed complexes; the observed dissociation rate constant was 3.2 x 10 (-4) s-1; and Ki increased to... WebbAdherence inhibition assays demonstrated varying degrees of disruption of the S. mutans-agglutinin interaction by anti-P1 monoclonal antibodies recognizing different epitopes, whereas a polyclonal reagent demonstrated more complete inhibition.
Inactivation of p27kip1 Promoted Nonspecific ... - Oxford Academic
Webb1 mars 2000 · The human glutathione transferase P1-1 specific inhibitor TER 117 designed for overcoming cytostatic-drug resistance is also a strong inhibitor of glyoxalase I. A. Johansson, M. Ridderström, B. Mannervik Published 1 March 2000 Biology, Chemistry Molecular pharmacology WebbThe cyclin-dependent kinase (Cdk) inhibitor p27 regulates cell proliferation, cell motility and apoptosis, and is inactivated through various means in many types of human cancer. Recent studies in ... death certificate dallas county
A whole cell BIAcore assay to evaluate P1-mediated adherence of ...
Webb6 feb. 1996 · However, the P1 (L)-proline analog 4a is a much poorer inhibitor of MMP-3 than is the phthalimide 3g. In addition, P1 (13)- and (L)-(N-acetyl)prolylaminobutyl analogs in a related series of phosphinic acid inhibitors were found to be equipotent, suggesting that the binding interactions in this region are largely hydrophobic and relatively … WebbDownload Table Selected X-ray and calculated bond angles (°) of inhibitor P1 from publication: Imidazo[4,5-b]pyridines as a New Class of Corrosion Inhibitors for Mild Steel: Experimental and ... Webb1 mars 1991 · Abstract. It has been shown that the P1 site (the center of the reactive site) of protease inhibitors corresponds to the specificity of the cognate protease, and consequently specificity of Streptomyces subtilisin inhibitor (SSI) can be altered by substitution of a single amino acid at the P1 site. In this paper, to investigate whether … generic bluetooth radio erro de driver